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Functional selectivity of GPCR-directed drug action through location bias

G protein-coupled receptors (GPCRs) are increasingly recognized to operate from intracellular membranes as well as the plasma membrane. The β(2)-adrenergic GPCR can activate Gs-linkedcyclic AMP (cAMP) signaling from endosomes. We show here that the homologous human β(1)-adrenergic receptor initiates...

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Bibliografiske detaljer
Udgivet i:Nat Chem Biol
Main Authors: Irannejad, Roshanak, Pessino, Veronica, Mika, Delphine, Huang, Bo, Wedegaertner, Philip B., Conti, Marco, von Zastrow, Mark
Format: Artigo
Sprog:Inglês
Udgivet: 2017
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5733145/
https://ncbi.nlm.nih.gov/pubmed/28553949
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.2389
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