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A facile cyclization method improves peptide serum stability and confers intrinsic fluorescence

Peptides are a growing class of macromolecules used in pharmaceutics. The path toward clinical use of candidate peptides involves sequence optimization and cyclization for stability and affinity. For internalized peptides, tagging is also often required for intracellular trafficking studies, althoug...

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Dettagli Bibliografici
Pubblicato in:Chembiochem
Autori principali: Ngambenjawong, Chayanon, Gustafson, Heather H., Sylvestre, Meilyn, Pun, Suzie H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5730504/
https://ncbi.nlm.nih.gov/pubmed/29044914
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201700446
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