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Site-Specific Radiofluorination of Biomolecules with 8-[(18)F]-Fluorooctanoic Acid Catalyzed by Lipoic Acid Ligase

New methodologies for site-specifically radiolabeling proteins with (18)F are required to generate high quality radiotracers for preclinical and clinical applications with positron emission tomography. Herein, we report an approach by which we use lipoic acid ligase (LplA) to conjugate [(18)F]-fluor...

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Detalhes bibliográficos
Publicado no:ACS Chem Biol
Main Authors: Drake, Christopher R., Sevillano, Natalia, Truillet, Charles, Craik, Charles S., VanBrocklin, Henry F., Evans, Michael J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5712215/
https://ncbi.nlm.nih.gov/pubmed/27008570
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.6b00172
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