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Phenolic Hydrazones are Potent Inhibitors of Macrophage Migration Inhibitory Factor Proinflammatory Activity and Survival Improving Agents in Sepsis()

A series of phenolic hydrazones were synthesized and evaluated for their inhibition of MIF tautomerase activity. Compound 7 emerged as a potent inhibitor of MIF with an IC(50) of 130 nM. Compound 7 dose dependently suppressed TNFα secretion from lipopolysaccharide stimulated macrophages. The therape...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Dabideen, Darrin R., Cheng, Kai Fan, Aljabari, Bayan, Miller, Edmund J., Pavlov, Valentin A., Al-Abed, Yousef
Formato: Artigo
Idioma:Inglês
Publicado em: 2007
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5710735/
https://ncbi.nlm.nih.gov/pubmed/17385848
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm061477+
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