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Dermatologic side effects associated with the MEK 1/2 inhibitor selumetinib (AZD6244, ARRY-142886)

BACKGROUND: Selumetinib (AZD6244, ARRY-142886) is a second generation MEK inhibitor that is currently in clinical trials for various solid malignancies. MEK kinase inhibitors are associated with dermatologic toxicities. While reactions affecting the skin, hair and nails to other targeted agents, suc...

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Dettagli Bibliografici
Pubblicato in:Invest New Drugs
Autori principali: Balagula, Yevgeniy, Barth, Katherine, Busam, Klaus J., Lacouture, Mario E., Chapman, Paul B., Myskowski, Patricia L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2010
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5691597/
https://ncbi.nlm.nih.gov/pubmed/20978926
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10637-010-9567-3
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