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The Therapeutic Antibody LM609 Selectively Inhibits Ligand Binding to Human α(V)β(3) Integrin via Steric Hindrance

The LM609 antibody specifically recognizes α(V)β(3) integrin and inhibits angiogenesis, bone resorption, and viral infections in an arginine-glycine-aspartate independent manner. LM609 entered phase II clinical trials for the treatment of several cancers and was also used for α(V)β(3)-targeted radio...

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Dettagli Bibliografici
Pubblicato in:Structure
Autori principali: Borst, Andrew J., James, Zachary M., Zagotta, William N., Ginsberg, Mark, Rey, Felix A., DiMaio, Frank, Backovic, Marija, Veesler, David
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5689087/
https://ncbi.nlm.nih.gov/pubmed/29033288
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.str.2017.09.007
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