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Role of P-Glycoprotein Inhibitors in the Bioavailability Enhancement of Solid Dispersion of Darunavir

OBJECTIVE: The aim of the present study was to improve bioavailability of an important antiretroviral drug, Darunavir (DRV), which has low water solubility and poor intestinal absorption through solid dispersion (SD) approach incorporating polymer with P-glycoprotein inhibitory potential. METHODS: A...

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Detaylı Bibliyografya
Yayımlandı:Biomed Res Int
Asıl Yazarlar: Rehman, Saleha, Nabi, Bushra, Fazil, Mohammad, Khan, Saba, Bari, Naimat Kalim, Singh, Romi, Ahmad, Shavej, Kumar, Varinder, Baboota, Sanjula, Ali, Javed
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Hindawi 2017
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC5684613/
https://ncbi.nlm.nih.gov/pubmed/29226149
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1155/2017/8274927
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