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Alkynyl Thioethers in Gold‐Catalyzed Annulations To Form Oxazoles

Non‐oxidative, regioselective, and convergent access to densely functionalized oxazoles is realized in a functional‐group tolerant manner using alkynyl thioethers. Sulfur‐terminated alkynes provide access to reactivity previously requiring strong donor‐substituted alkynes such as ynamides. Sulfur do...

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Publicado en:Angew Chem Int Ed Engl
Autores principales: Reddy, Raju Jannapu, Ball‐Jones, Matthew P., Davies, Paul W.
Formato: Artigo
Lenguaje:Inglês
Publicado: John Wiley and Sons Inc. 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5656920/
https://ncbi.nlm.nih.gov/pubmed/28841255
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201706850
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