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The drug transporter OAT3 (SLC22A8) and endogenous metabolite communication via the gut–liver–kidney axis

The organic anion transporters OAT1 (SLC22A6) and OAT3 (SLC22A8) have similar substrate specificity for drugs, but it is far from clear whether this holds for endogenous substrates. By analysis of more than 600 metabolites in the Oat3KO (Oat3 knockout) by LC/MS, we demonstrate OAT3 involvement in th...

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Pubblicato in:J Biol Chem
Autori principali: Bush, Kevin T., Wu, Wei, Lun, Christina, Nigam, Sanjay K.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5612110/
https://ncbi.nlm.nih.gov/pubmed/28765282
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M117.796516
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