Načítá se...

Paralog-divergent Features May Help Reduce Off-target Effects of Drugs: Hints from Glucagon Subfamily Analysis

Side effects from targeted drugs remain a serious concern. One reason is the nonselective binding of a drug to unintended proteins such as its paralogs, which are highly homologous in sequences and have similar structures and drug-binding pockets. To identify targetable differences between paralogs,...

Celý popis

Uloženo v:
Podrobná bibliografie
Vydáno v:Genomics Proteomics Bioinformatics
Hlavní autoři: Sa, Zhining, Zhou, Jingqi, Zou, Yangyun, Su, Zhixi, Gu, Xun
Médium: Artigo
Jazyk:Inglês
Vydáno: Elsevier 2017
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5582795/
https://ncbi.nlm.nih.gov/pubmed/28642113
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.gpb.2017.03.004
Tagy: Přidat tag
Žádné tagy, Buďte první, kdo otaguje tento záznam!