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[(3)H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors

MRS 1754 [N-(4-cyanophenyl)-2-[4-(2,3,6,7-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)-phenoxy]acetamide] is a selective antagonist ligand of A(2B) adenosine receptors. This is the least well-defined adenosine receptor subtype, and A(2B) antagonists have potential as antiasthmatic drugs. For use...

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Detalhes bibliográficos
Publicado no:Biochem Pharmacol
Main Authors: Ji, Xiao-duo, Kim, Yong-Chul, Ahern, David G., Linden, Joel, Jacobson, Kenneth A.
Formato: Artigo
Idioma:Inglês
Publicado em: 2001
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5567772/
https://ncbi.nlm.nih.gov/pubmed/11266650
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