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Testing inhomogeneous solvation theory in structure-based ligand discovery

Binding-site water is often displaced upon ligand recognition, but is commonly neglected in structure-based ligand discovery. Inhomogeneous solvation theory (IST) has become popular for treating this effect, but it has not been tested in controlled experiments at atomic resolution. To do so, we turn...

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Detalles Bibliográficos
Publicado en:Proc Natl Acad Sci U S A
Main Authors: Balius, Trent E., Fischer, Marcus, Stein, Reed M., Adler, Thomas B., Nguyen, Crystal N., Cruz, Anthony, Gilson, Michael K., Kurtzman, Tom, Shoichet, Brian K.
Formato: Artigo
Idioma:Inglês
Publicado: National Academy of Sciences 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5565424/
https://ncbi.nlm.nih.gov/pubmed/28760952
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1703287114
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