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Inhibition of Sodium Ion Channel Function with Truncated Forms of Batrachotoxin

A novel family of small molecule inhibitors of voltage-gated sodium channels (Na(v)s) based on the structure of batrachotoxin (BTX) – a well-known channel agonist – is described. Protein mutagenesis and electrophysiology experiments reveal the binding site as the inner pore region of the channel, an...

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Publicado en:ACS Chem Neurosci
Main Authors: Toma, Tatsuya, Logan, Matthew M., Menard, Frederic, Devlin, A. Sloan, Bois, J. Du
Formato: Artigo
Idioma:Inglês
Publicado: 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5555364/
https://ncbi.nlm.nih.gov/pubmed/27501251
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.6b00212
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