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TKI-addicted ROS1-rearranged cells are destined to survival or death by the intensity of ROS1 kinase activity

ROS1 rearrangement is observed in 1–2% of non-small cell lung cancers (NSCLC). The ROS1 tyrosine kinase inhibitor (TKI) crizotinib has induced marked tumour shrinkage in ROS1-rearranged cancers. However, emergence of acquired resistance to TKI is inevitable within a few years. Previous findings indi...

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Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Ogura, Hayato, Nagatake-Kobayashi, Yuka, Adachi, Jun, Tomonaga, Takeshi, Fujita, Naoya, Katayama, Ryohei
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5514057/
https://ncbi.nlm.nih.gov/pubmed/28717217
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-05736-9
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