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Virtual Screening, pharmacophore development and structure based similarity search to identify inhibitors against IdeR, a transcription factor of Mycobacterium tuberculosis

ideR, an essential gene of Mycobacterium tuberculosis, is an attractive drug target as its conditional knockout displayed attenuated growth phenotype in vitro and in vivo. To the best of our knowledge, no inhibitors of IdeR are identified. We carried out virtual screening of NCI database against the...

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Publicado en:Sci Rep
Main Authors: Rohilla, Akshay, Khare, Garima, Tyagi, Anil K.
Formato: Artigo
Idioma:Inglês
Publicado: Nature Publishing Group UK 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5498548/
https://ncbi.nlm.nih.gov/pubmed/28680150
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-04748-9
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