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Dynamical models of mutated chronic myelogenous leukemia cells for a post-imatinib treatment scenario: Response to dasatinib or nilotinib therapy

Targeted inhibition of the oncogenic BCR-ABL1 fusion protein using the ABL1 tyrosine kinase inhibitor imatinib has become standard therapy for chronic myelogenous leukemia (CML), with most patients reaching total and durable remission. However, a significant fraction of patients develop resistance,...

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Библиографические подробности
Опубликовано в: :PLoS One
Главные авторы: Woywod, Clemens, Gruber, Franz X., Engh, Richard A., Flå, Tor
Формат: Artigo
Язык:Inglês
Опубликовано: Public Library of Science 2017
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5497988/
https://ncbi.nlm.nih.gov/pubmed/28678800
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0179700
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