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Rucaparib: the past, present, and future of a newly approved PARP inhibitor for ovarian cancer

Rucaparib camsylate (CO-338, AG-014699, PF-01367338) is a potent PARP-1, PARP-2, and PARP-3 inhibitor. Phase I and II studies demonstrated clinical efficacy in both BRCA-mutated (inclusive of germline and somatic) ovarian tumors and ovarian tumors with homologous recombination deficiency (HRD) loss...

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Pubblicato in:Onco Targets Ther
Autori principali: Dockery, LE, Gunderson, CC, Moore, KN
Natura: Artigo
Lingua:Inglês
Pubblicazione: Dove Medical Press 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5488752/
https://ncbi.nlm.nih.gov/pubmed/28790837
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/OTT.S114714
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