A carregar...

Evaluation of rucaparib and companion diagnostics in the PARP inhibitor landscape for recurrent ovarian cancer therapy

Rucaparib camsylate (CO-338; 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one ((1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]hept-1-yl)methanesulfonic acid salt) is a PARP1, 2 and 3 inhibitor. Phase I studies identified a recommended Phase II dose of 600 mg ora...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Future Oncol
Main Authors: Jenner, Zachary B, Sood, Anil K, Coleman, Robert L
Formato: Artigo
Idioma:Inglês
Publicado em: Future Medicine Ltd 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4976841/
https://ncbi.nlm.nih.gov/pubmed/27087632
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2217/fon-2016-0002
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!