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Should Low Molecular Weight PSMA Targeted Ligands Get Bigger and Use Albumin Ligands for PSMA Targeting?

Prostate Specific Membrane Antigen (PSMA) is strongly expressed in prostate cancer. Recently a number of low-molecular-weight inhibitors have demonstrated excellent PSMA targeting activity for both imaging as well as Lutecium-177 radiotherapy in human trials. The paper by Choy et al raises the quest...

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Publicat a:Theranostics
Autors principals: Huang, Steve S., Heston, Warren D.W.
Format: Artigo
Idioma:Inglês
Publicat: Ivyspring International Publisher 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5479280/
https://ncbi.nlm.nih.gov/pubmed/28638479
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.7150/thno.20284
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