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Inhibition of PDE5A1 guanosine cyclic monophosphate (cGMP) hydrolysing activity by sildenafil analogues that inhibit cellular cGMP efflux

OBJECTIVES: To determine the ability of 11 sildenafil analogues to discriminate between cyclic nucleotide phosphodiesterases (cnPDEs) and to characterise their inhibitory potencies (K (i) values) of PDE5A1‐dependent guanosine cyclic monophosphate (cGMP) hydrolysis. METHODS: Sildenafil analogues were...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:J Pharm Pharmacol
Hauptverfasser: Subbotina, Anna, Ravna, Aina W., Lysaa, Roy A., Abagyan, Ruben, Bugno, Ryszard, Sager, Georg
Format: Artigo
Sprache:Inglês
Veröffentlicht: John Wiley and Sons Inc. 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5434896/
https://ncbi.nlm.nih.gov/pubmed/28211580
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/jphp.12693
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