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Metabolic Profiles of Pomalidomide in Human Plasma Simulated with Pharmacokinetic Data in Control and Humanized-liver Mice

1. Pomalidomide has been shown to be potentially teratogenic in thalidomide-sensitive animal species such as rabbits. Screening for thalidomide analogs devoid of teratogenicity/toxicity—attributable to metabolites formed by cytochrome P450 enzymes—but having immunomodulatory properties is a strategi...

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Dettagli Bibliografici
Pubblicato in:Xenobiotica
Autori principali: Shimizu, Makiko, Suemizu, Hiroshi, Mitsui, Marina, Shibata, Norio, Guengerich, F. Peter, Yamazaki, Hiroshi
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5433912/
https://ncbi.nlm.nih.gov/pubmed/27852146
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/00498254.2016.1247218
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