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Unique residues in the ATP gated human P2X7 receptor define a novel allosteric binding pocket for the selective antagonist AZ10606120

The P2X7 receptor (P2X7R) for ATP is a therapeutic target for pathophysiological states including inflammation, pain management and epilepsy. This is facilitated by the predicted low side effect profile as the high concentrations of ATP required to activate the receptor are usually only found follow...

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Bibliografske podrobnosti
izdano v:Sci Rep
Main Authors: Allsopp, Rebecca C., Dayl, Sudad, Schmid, Ralf, Evans, Richard J.
Format: Artigo
Jezik:Inglês
Izdano: Nature Publishing Group UK 2017
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5429621/
https://ncbi.nlm.nih.gov/pubmed/28389651
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-00732-5
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