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Optimization of intestinal microsomal preparation in the rat: A systematic approach to assess the influence of various methodologies on metabolic activity and scaling factors

The metabolic capacity of the intestine and its importance as the initial barrier to systemic exposure can lead to underestimation of first‐pass, and thus overestimation of oral bioavailability. However, the in vitro tools informing estimates of in vivo intestinal metabolism are limited by the compl...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Biopharm Drug Dispos
Hauptverfasser: Hatley, Oliver J.D., Jones, Christopher R., Galetin, Aleksandra, Rostami‐Hodjegan, Amin
Format: Artigo
Sprache:Inglês
Veröffentlicht: John Wiley and Sons Inc. 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5413848/
https://ncbi.nlm.nih.gov/pubmed/28207929
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/bdd.2070
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