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Targeting MYC Dependence by Metabolic Inhibitors in Cancer

MYC is a critical growth regulatory gene that is commonly overexpressed in a wide range of cancers. Therapeutic targeting of MYC transcriptional activity has long been a goal, but it has been difficult to achieve with drugs that directly block its DNA-binding ability. Additional approaches that expl...

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Dettagli Bibliografici
Pubblicato in:Genes (Basel)
Autori principali: Sabnis, Himalee S., Somasagara, Ranganatha R., Bunting, Kevin D.
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5406861/
https://ncbi.nlm.nih.gov/pubmed/28362357
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/genes8040114
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