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AEE788 Inhibits Basal Body Assembly and Blocks DNA Replication in the African Trypanosome

Trypanosoma brucei causes human African trypanosomiasis (HAT). The pyrrolopyrimidine AEE788 (a hit for anti-HAT drug discovery) associates with three trypanosome protein kinases. Herein we delineate the effects of AEE788 on T. brucei using chemical biology strategies. AEE788 treatment inhibits DNA r...

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Dettagli Bibliografici
Pubblicato in:Mol Pharmacol
Autori principali: Sullenberger, Catherine, Piqué, Daniel, Ogata, Yuko, Mensa-Wilmot, Kojo
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5399642/
https://ncbi.nlm.nih.gov/pubmed/28246189
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.116.106906
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