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K+ channel openers activate brain sulfonylurea-sensitive K+ channels and block neurosecretion.

Vascular K+ channel openers such as cromakalim, nicorandil, and pinacidil potently stimulate 86Rb+ efflux from slices of substantia nigra. This 86Rb+ efflux is blocked by antidiabetic sulfonylureas, which are known to be potent and specific blockers of ATP-regulated K+ channels in pancreatic beta ce...

Täydet tiedot

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Bibliografiset tiedot
Päätekijät: Schmid-Antomarchi, H, Amoroso, S, Fosset, M, Lazdunski, M
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 1990
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC53926/
https://ncbi.nlm.nih.gov/pubmed/2333295
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