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Structural features embedded in G protein-coupled receptor co-crystal structures are key to their success in virtual screening

Structure based drug discovery on GPCRs harness atomic detail X-ray binding pockets and large libraries of potential drug lead candidates in virtual screening (VS) to identify novel lead candidates. Relatively small conformational differences between such binding pockets can be critical to the succe...

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Pubblicato in:PLoS One
Autori principali: Coudrat, Thomas, Christopoulos, Arthur, Sexton, Patrick Michael, Wootten, Denise
Natura: Artigo
Lingua:Inglês
Pubblicazione: Public Library of Science 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5381884/
https://ncbi.nlm.nih.gov/pubmed/28380046
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0174719
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