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In silico discovery and in vitro activity of inhibitors against Mycobacterium tuberculosis 7,8-diaminopelargonic acid synthase (Mtb BioA)

Computer-aided drug discovery and development approaches such as virtual screening, molecular docking, and in silico drug property calculations have been utilized in this effort to discover new lead compounds against tuberculosis. The enzyme 7,8-diaminopelargonic acid aminotransferase (BioA) in Myco...

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Detalles Bibliográficos
Publicado en:Drug Des Devel Ther
Autores principales: Billones, Junie B, Carrillo, Maria Constancia O, Organo, Voltaire G, Sy, Jamie Bernadette A, Clavio, Nina Abigail B, Macalino, Stephani Joy Y, Emnacen, Inno A, Lee, Alexandra P, Ko, Paul Kenny L, Concepcion, Gisela P
Formato: Artigo
Lenguaje:Inglês
Publicado: Dove Medical Press 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5338852/
https://ncbi.nlm.nih.gov/pubmed/28280303
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/DDDT.S119930
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