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Design, Synthesis, and Biological Evaluation of Potential Prodrugs Related to the Experimental Anticancer Agent Indotecan (LMP400)

Indenoisoquinoline topoisomerase I (Top1) inhibitors are a novel class of anticancer agents with two compounds in clinical trials. Recent metabolism studies of indotecan (LMP400) led to the discovery of the biologically active 2-hydroxylated analogue and 3-hydroxylated metabolite, thus providing str...

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Bibliographic Details
Published in:J Med Chem
Main Authors: Lv, Peng-Cheng, Elsayed, Mohamed S. A., Agama, Keli, Marchand, Christophe, Pommier, Yves, Cushman, Mark
Format: Artigo
Language:Inglês
Published: 2016
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC5317102/
https://ncbi.nlm.nih.gov/pubmed/27097152
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b00220
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