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Cell-intrinsic determinants of ibrutinib-induced apoptosis in Chronic Lymphocytic Leukemia

PURPOSE: Ibrutinib, a Bruton’s tyrosine kinase (BTK) inhibitor, is approved for the treatment of relapsed CLL and CLL with del17p. Mechanistically, ibrutinib interferes with BCR signaling as well as multiple CLL cell to microenvironment interactions. Given the importance of ibrutinib in the manageme...

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Publicat a:Clin Cancer Res
Autors principals: Amin, Nisar A., Balasubramanian, Sriram, Saiya-Cork, Kamlai, Shedden, Kerby, Hu, Nan, Malek, Sami N.
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5315657/
https://ncbi.nlm.nih.gov/pubmed/27535981
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-15-2921
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