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Bazedoxifene as a Novel GP130 Inhibitor for Pancreatic Cancer Therapy

The IL-6/GP130/STAT3 pathway is crucial for tumorigenesis in multiple cancer types, including pancreatic cancer and presents as a viable target for cancer therapy. We reported Bazedoxifene, which is approved as a selective estrogen modulator by FDA, as a novel inhibitor of IL-6/GP130 protein−protein...

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Publicat a:Mol Cancer Ther
Autors principals: Wu, Xiaojuan, Cao, Yang, Xiao, Hui, Li, Chenglong, Lin, Jiayuh
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5310670/
https://ncbi.nlm.nih.gov/pubmed/27535971
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1535-7163.MCT-15-0921
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