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Molecular Pathways: Maintaining MAPK inhibitor sensitivity by targeting non-mutational tolerance

Targeting hyperactive MAPK signaling has proven to be an effective treatment for a variety of different cancers. Responses to the BARF inhibitors vemurafenib or dabrafenib and MEK inhibitors trametinib or cobimentinib are however transient and complete remission is rarely observed; rather outgrowth...

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Bibliografski detalji
Izdano u:Clin Cancer Res
Glavni autori: Smith, Michael P, Wellbrock, Claudia
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5300098/
https://ncbi.nlm.nih.gov/pubmed/27797970
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-16-0954
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