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Griseofulvin impairs intraerythrocytic growth of Plasmodium falciparum through ferrochelatase inhibition but lacks activity in an experimental human infection study

Griseofulvin, an orally active antifungal drug used to treat dermatophyte infections, has a secondary effect of inducing cytochrome P450-mediated production of N-methyl protoporphyrin IX (N-MPP). N-MPP is a potent competitive inhibitor of the heme biosynthetic-enzyme ferrochelatase, and inhibits the...

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書目詳細資料
發表在:Sci Rep
Main Authors: Smith, Clare M., Jerkovic, Ante, Truong, Thy Thuc, Foote, Simon J., McCarthy, James S., McMorran, Brendan J.
格式: Artigo
語言:Inglês
出版: Nature Publishing Group 2017
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC5296727/
https://ncbi.nlm.nih.gov/pubmed/28176804
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep41975
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