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Efavirenz Is Predicted To Accumulate in Brain Tissue: an In Silico, In Vitro, and In Vivo Investigation

Adequate concentrations of efavirenz in the central nervous system (CNS) are necessary to suppress viral replication, but high concentrations may increase the likelihood of CNS adverse drug reactions. The aim of this investigation was to evaluate the efavirenz distribution in the cerebrospinal fluid...

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Publicado en:Antimicrob Agents Chemother
Autores principales: Curley, Paul, Rajoli, Rajith K. R., Moss, Darren M., Liptrott, Neill J., Letendre, Scott, Owen, Andrew, Siccardi, Marco
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Microbiology 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5192136/
https://ncbi.nlm.nih.gov/pubmed/27799216
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01841-16
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