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Therapeutic potential of JAK2 inhibitors

The discovery of an activating tyrosine kinase mutation JAK2V617F in myeloproliferative neoplasms (MPNs), polycythemia vera (PV), essential thrombocythemia (ET) and primary myelofibrosis (PMF) has resulted in the development of JAK2 inhibitors, of which several are being evaluated in phase I/II clin...

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Publicat a:Hematology Am Soc Hematol Educ Program
Autor principal: Verstovsek, Srdan
Format: Artigo
Idioma:Inglês
Publicat: 2009
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5166576/
https://ncbi.nlm.nih.gov/pubmed/20008249
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/asheducation-2009.1.636
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