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Dual activities of ritanserin and R59022 as DGKα inhibitors and serotonin receptor antagonists

Diacylglycerol kinase alpha (DGKα) catalyzes the conversion of diacylglycerol (DAG) to phosphatidic acid (PA). Recently, DGKα was identified as a therapeutic target in various cancers, as well as in immunotherapy. Application of small-molecule DGK inhibitors, R59022 and R59949, induces cancer cell d...

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Detaylı Bibliyografya
Yayımlandı:Biochem Pharmacol
Asıl Yazarlar: Boroda, Salome, Niccum, Maria, Raje, Vidisha, Purow, Benjamin W., Harris, Thurl E.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2016
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC5164959/
https://ncbi.nlm.nih.gov/pubmed/27974147
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2016.10.011
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