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Lipid-modified G4-decoy oligonucleotide anchored to nanoparticles: delivery and bioactivity in pancreatic cancer cells

KRAS is mutated in >90% of pancreatic ductal adenocarcinomas. As its inactivation leads to tumour regression, mutant KRAS is considered an attractive target for anticancer drugs. In this study we report a new delivery strategy for a G4-decoy oligonucleotide that sequesters MAZ, a transcription fa...

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Détails bibliographiques
Publié dans:Sci Rep
Auteurs principaux: Cogoi, S., Jakobsen, U., Pedersen, E. B., Vogel, S., Xodo, L. E.
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group 2016
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5144097/
https://ncbi.nlm.nih.gov/pubmed/27929127
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep38468
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