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Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Arginases are enzymes that are involved in many human diseases and have been targeted for new treatments. Here a series of cinnamides was designed, synthesized and evaluated in vitro and in silico for their inhibitory activity against mammalian arginase. Using a microassay on purified liver bovine a...

詳細記述

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書誌詳細
出版年:Int J Mol Sci
主要な著者: Pham, Thanh-Nhat, Bordage, Simon, Pudlo, Marc, Demougeot, Céline, Thai, Khac-Minh, Girard-Thernier, Corine
フォーマット: Artigo
言語:Inglês
出版事項: MDPI 2016
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC5085689/
https://ncbi.nlm.nih.gov/pubmed/27690022
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms17101656
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