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The PARP inhibitor ABT-888 potentiates darbazine-induced cell death in carcinoids

Monoagent DNA-alkylating chemotherapies like dacarbazine are among a paucity of medical treatments for advanced carcinoid tumors, but are limited by host toxicity and intrinsic chemoresistance through the base excision repair (BER) pathway via poly (ADP-ribose) polymerase (PARP). Hence, inhibitors o...

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Dades bibliogràfiques
Publicat a:Cancer Gene Ther
Autors principals: Somnay, Yash, Lubner, Sam, Gill, Harpreet, Matsumura, Jon Blake, Chen, Herbert
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5083201/
https://ncbi.nlm.nih.gov/pubmed/27632933
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/cgt.2016.39
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