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Synthesis and NMR studies of malonyl-linked glycoconjugates of N-(2-aminoethyl)glycine. Building blocks for the construction of combinatorial glycopeptide libraries

Four glycoconjugate building blocks for the construction of combinatorial PNA like glycopeptide libraries were prepared in 75–79% yield by condensing tert-butyl N-[2-(N-9-fluorenylmethoxycarbonylamino)ethyl]glycinate (AEG) 5 with 3-oxo-3-(2,3,4,6-tetra-O-acetyl-β-D-glucopyranosylamino)- (6a), 3-oxo-...

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Pubblicato in:Beilstein J Org Chem
Autori principali: Nörrlinger, Markus, Hafner, Sven, Ziegler, Thomas
Natura: Artigo
Lingua:Inglês
Pubblicazione: Beilstein-Institut 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5082468/
https://ncbi.nlm.nih.gov/pubmed/27829900
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.12.183
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