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Inhibitory Interaction Potential of 22 Antituberculosis Drugs on Organic Anion and Cation Transporters of the SLC22A Family

Twenty-two currently marketed antituberculosis drugs were comprehensively evaluated for their inhibitory effect on organic anionic transporter (OAT)- and organic cation transporter (OCT)-mediated uptake using stably transfected HEK293 cells in vitro. We observed moderate to strong inhibitory effects...

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Détails bibliographiques
Publié dans:Antimicrob Agents Chemother
Auteurs principaux: Parvez, M. Masud, Kaisar, Nazia, Shin, Ho Jung, Jung, Jin Ah, Shin, Jae-Gook
Format: Artigo
Langue:Inglês
Publié: American Society for Microbiology 2016
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5075059/
https://ncbi.nlm.nih.gov/pubmed/27550354
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01151-16
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