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EZH2 inhibitors transcriptionally upregulate cytotoxic autophagy and cytoprotective unfolded protein response in human colorectal cancer cells

Enhancer of zeste homolog 2 (EZH2) has been emerged as novel anticancer target. Various EZH2 small-molecule inhibitors have been developed in recent years. A major class of EZH2 inhibitors are S-adenosyl-L-methionine (SAM)-competitive inhibitors, such as EPZ005687, EI1, GSK126, UNC1999 and GSK343. A...

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Bibliografski detalji
Izdano u:Am J Cancer Res
Glavni autori: Hsieh, Yao-Yu, Lo, Hsiang-Ling, Yang, Pei-Ming
Format: Artigo
Jezik:Inglês
Izdano: e-Century Publishing Corporation 2016
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Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5004071/
https://ncbi.nlm.nih.gov/pubmed/27648357
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