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Structural Basis of Microtubule Destabilization by Potent Auristatin Anti-Mitotics

The auristatin class of microtubule destabilizers are highly potent cytotoxic agents against several cancer cell types when delivered as antibody drug conjugates. Here we describe the high resolution structures of tubulin in complex with both monomethyl auristatin E and F and unambiguously define th...

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Dettagli Bibliografici
Pubblicato in:PLoS One
Autori principali: Waight, Andrew B., Bargsten, Katja, Doronina, Svetlana, Steinmetz, Michel O., Sussman, Django, Prota, Andrea E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Public Library of Science 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4982639/
https://ncbi.nlm.nih.gov/pubmed/27518442
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0160890
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