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A novel bis(pinacolato)diboron-mediated N–O bond deoxygenative route to C6 benzotriazolyl purine nucleoside derivatives()

Reaction of amide bonds in t-butyldimethylsilyl-protected inosine, 2′-deoxyinosine, guanosine, 2′-deoxyguanosine, and 2-phenylinosine with commercially available peptide-coupling agents (benzotriazol-1H-yloxy)tris(dimethylaminophosphonium) hexafluorophosphate (BOP), (6-chloro-benzotriazol-1H-yloxy)t...

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Publicat a:Org Biomol Chem
Autors principals: Basava, Vikram, Yang, Lijia, Pradhan, Padmanava, Lakshman, Mahesh K.
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4981646/
https://ncbi.nlm.nih.gov/pubmed/27377367
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6ob01170e
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