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Novel ligands of Choline Acetyltransferase designed by in silico molecular docking, hologram QSAR and lead optimization

Recent reports have brought back the acetylcholine synthesizing enzyme, choline acetyltransferase in the mainstream research in dementia and the cholinergic anti-inflammatory pathway. Here we report, a specific strategy for the design of novel ChAT ligands based on molecular docking, Hologram Quanti...

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Detaylı Bibliyografya
Yayımlandı:Sci Rep
Asıl Yazarlar: Kumar, Rajnish, Långström, Bengt, Darreh-Shori, Taher
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Nature Publishing Group 2016
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4978996/
https://ncbi.nlm.nih.gov/pubmed/27507101
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep31247
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