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Ergosterol-loaded poly(lactide-co-glycolide) nanoparticles with enhanced in vitro antitumor activity and oral bioavailability

AIM: Ergosterol is a plant sterol with anti-tumor and anti-angiogenic activities, but is poorly soluble. In this study, we attempted to enhance its anti-tumor action and oral bioavailability via poly(lactide-co-glycolide) (PLGA) nanoparticle encapsulation. METHODS: Ergosterol-loaded PLGA nanoparticl...

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Detalhes bibliográficos
Publicado no:Acta Pharmacol Sin
Main Authors: Zhang, Hui-yun, Firempong, Caleb Kesse, Wang, Yuan-wen, Xu, Wen-qian, Wang, Miao-miao, Cao, Xia, Zhu, Yuan, Tong, Shan-shan, Yu, Jiang-nan, Xu, Xi-ming
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2016
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4954769/
https://ncbi.nlm.nih.gov/pubmed/27133301
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/aps.2016.37
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