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Ligand Docking to Intermediate and Close-To-Bound Conformers Generated by an Elastic Network Model Based Algorithm for Highly Flexible Proteins

Incorporating receptor flexibility in small ligand-protein docking still poses a challenge for proteins undergoing large conformational changes. In the absence of bound structures, sampling conformers that are accessible by apo state may facilitate docking and drug design studies. For this aim, we d...

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Detalhes bibliográficos
Publicado no:PLoS One
Main Authors: Kurkcuoglu, Zeynep, Doruker, Pemra
Formato: Artigo
Idioma:Inglês
Publicado em: Public Library of Science 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4922591/
https://ncbi.nlm.nih.gov/pubmed/27348230
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0158063
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