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DRUG EVALUATION: Pharmacodynamic assessment of vedolizumab for the treatment of ulcerative colitis

INTRODUCTION: Vedolizumab is an anti-integrin approved for the treatment of Crohn’s disease and ulcerative colitis. By binding the α4β7-integrin heterodimer, vedolizumab blocks leukocyte translocation into gastrointestinal tissue. AREAS COVERED: This review discusses the chemistry, pharmacologic pro...

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Publicat a:Expert Opin Drug Metab Toxicol
Autors principals: McLean, Leon P., Cross, Raymond K.
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4917449/
https://ncbi.nlm.nih.gov/pubmed/27096357
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/17425255.2016.1181171
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