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A new autoinhibited kinase conformation reveals a salt-bridge switch in kinase activation

In the structure of autoinhibited EphA2 tyrosine kinase reported herein, we have captured the entire activation segment, revealing a previously unknown role of the conserved Arg762 in kinase autoinhibition by interacting with the essential Mg(2+)-chelating Asp757. While it is well known that this Ar...

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Bibliografiske detaljer
Udgivet i:Sci Rep
Main Authors: Wei, Qiang, Yang, Shaoyuan, Li, Dan, Zhang, Xiaoying, Zheng, Jimin, Jia, Zongchao
Format: Artigo
Sprog:Inglês
Udgivet: Nature Publishing Group 2016
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4914941/
https://ncbi.nlm.nih.gov/pubmed/27324091
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep28437
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