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Tissue barriers and novel approaches to achieve hepatoselectivity of subcutaneously-injected insulin therapeutics

Current subcutaneously (s.c.)-injected insulin (INS) products result in a hyperinsulin exposure to peripheral tissues (skeletal muscle and adipose) while INS hardly accesses to liver after injection. This unphysiological distribution raises risks of hypoglycemia episode and causes weight gain after...

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Pubblicato in:Tissue Barriers
Autori principali: Shao, Juntang, Zaro, Jennica L., Shen, Wei-Chiang
Natura: Artigo
Lingua:Inglês
Pubblicazione: Taylor & Francis 2016
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4910833/
https://ncbi.nlm.nih.gov/pubmed/27358753
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/21688370.2016.1156804
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